Taltirelin acetate

CAS No. 1549593-23-8

Taltirelin acetate ( TA-0910 acetate )

Catalog No. M22365 CAS No. 1549593-23-8

Taltirelin acetate is a superagonist at thyrotropin-releasing hormone receptor (TRH-R)(IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release)).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 42 Get Quote
10MG 69 Get Quote
25MG 143 Get Quote
50MG 284 Get Quote
100MG 510 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    Taltirelin acetate
  • Note
    Research use only, not for human use.
  • Brief Description
    Taltirelin acetate is a superagonist at thyrotropin-releasing hormone receptor (TRH-R)(IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release)).
  • Description
    Taltirelin acetate is a superagonist at thyrotropin-releasing hormone receptor (TRH-R)(IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release)).
  • Synonyms
    TA-0910 acetate
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    THR
  • Research Area
    Nervous system
  • Indication
    Spinocerebellar Degeneration

Chemical Information

  • CAS Number
    1549593-23-8
  • Formula Weight
    465.46
  • Molecular Formula
    C19H27N7O7
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:125 mg/mL (268.55 mM; Need ultrasonic)
  • SMILES
    O=C(N(CCC1)[C@@H]1C(N)=O)[C@@H](NC([C@@H](NC2=O)CC(N2C)=O)=O)CC3=CN=CN3.CC(O)=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Thirunarayanan N, et al. Taltirelin is a superagonist at the human thyrotropin-releasing hormone receptor. Front Endocrinol (Lausanne). 2012 Oct 9;3:120.
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